Nghiên cứu tổng hợp và đánh giá hoạt tính gây độc tế bào các dẫn xuất của benzimidazole và indole - 23

108. S. Bansal, S. Sur and V. Tandon, Benzimidazoles: Selective inhibitors of topoisomerase I with differential modes of action, Biochemistry, 2018, 58 (6), 809-817.

109. J. S. Kim, Q. Sun, B. Gatto, C. Yu, A. Liu, L. F. Liu and E. J. LaVoie, Structure-activity relationships of benzimidazoles and related heterocycles as topoisomerase I poisons, Bioorg. Med. Chem., 1996, 4 (4), 621-630.

110. A. S. Alpan, H. S. Gunes and Z. Topcu, 1H-Benzimidazole derivatives as mammalian DNA topoisomerase I inhibitors, Acta Biochim. Pol., 2007, 54 (3), 561-565.

111. U. Issar, R. Arora, T. Kumari and R. Kakkar, Combined pharmacophore- guided 3D-QSAR, molecular docking, and virtual screening on bis- benzimidazoles and ter-benzimidazoles as DNA–topoisomerase I poisons, Struct. Chem., 2019, 30 (4), 1185-1201.

112. A. L.-F. Chan, W.-S. Chang, L.-M. Chen, C.-M. Lee, C.-E. Chen, C.-M. Lin and J.-L. Hwang, Evodiamine stabilizes topoisomerase I-DNA cleavable complex to inhibit topoisomerase I activity, Molecules, 2009, 14 (4), 1342- 1352.

113. R. Chaniyara, S. Tala, C.-W. Chen, X. Zang, R. Kakadiya, L.-F. Lin, C.-H. Chen, S.-I. Chien, T.-C. Chou and T.-H. Tsai, Novel antitumor indolizino [6, 7-b] indoles with multiple modes of action: DNA cross-linking and topoisomerase I and II inhibition, J. Med. Chem., 2013, 56 (4), 1544-1563.

114. C. Zhang, Y. Qu and B. Niu, Design, synthesis and biological evaluation of lapachol derivatives possessing indole scaffolds as topoisomerase I inhibitors, Bioorg. Med. Chem., 2016, 24 (22), 5781-5786.

115. B. Shu, Q. Yu, D.-x. Hu, T. Che, S.-s. Zhang and D. Li, Synthesis and biological evaluation of novel indole-pyrazoline hybrid derivatives as potential topoisomerase 1 inhibitors, Bioorg. Med. Chem. Lett., 2020, 30 (4), 126925.

116. G. Dong, C. Sheng, S. Wang, Z. Miao, J. Yao and W. Zhang, Selection of evodiamine as a novel topoisomerase I inhibitor by structure-based virtual screening and hit optimization of evodiamine derivatives as antitumor agents, J. Med. Chem., 2010, 53 (21), 7521-7531.

117. B. Eren and Y. Bekdemir, Simple, mild, and highly efficient synthesis of 2- substituted benzimidazoles and bis-benzimidazoles, Quim. Nova, 2014, 37 (4), 643-647.

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118. U. C. Rajesh, R. Kholiya, V. S. Pavan and D. S. Rawat, Catalyst-free, ethylene glycol promoted one-pot three component synthesis of 3-amino alkylated indoles via Mannich-type reaction, Tetrahedron Lett., 2014, 55 (18), 2977- 2981.

119. A. Jindal and S. Vasudevan, Molecular Conformation and Hydrogen Bond Formation in Liquid Ethylene Glycol, J. Phys. Chem., 2020, 124 (41), 9136- 9143.

Nghiên cứu tổng hợp và đánh giá hoạt tính gây độc tế bào các dẫn xuất của benzimidazole và indole - 23

120. M. Krest’yaninov, A. Titova and A. Zaichikov, Intra-and intermolecular hydrogen bonds in ethylene glycol, monoethanolamine, and ethylenediamine, Russ. J. Phys. Chem., 2014, 88 (12), 2114-2120.

121. E. Chacon, D. Acosta and J. J. Lemasters, Primary cultures of cardiac myocytes as in vitro models for pharmacological and toxicological assessments, In Vitro Methods Pharm. Res., 1997, 209-223.

122. T. Mosmann, Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays, J. Immunol. Methods, 1983, 65 (1-2), 55-63.

123. ChemDraw 19.1, https://perkinelmer-chemscript- x64.software.informer.com/19.1/, truy cập ngày 22/5/2019.

124. Molecular operating environment (MOE) 2015.10,

https://www.chemcomp.com/Products.htm, truy cập ngày 18/10/2019.

125. Sybyl-X 1.1, https://sybyl-x.software.informer.com/1.1/, truy cập ngày 02/01/2020.

126. LeadIT 2.1. 8, https://www.biosolveit.de/LeadIT/, truy cập ngày 10/2/2020.

127. Discovery Studio Visualizer 4.0, https://discover.3ds.com/discovery-studio- visualizer-download, truy cập ngày 16/8/2020.

128. G. Navarrete‐Vázquez, H. Moreno‐Diaz, S. Estrada‐Soto, M. Torres‐Piedra, I. León‐Rivera, H. Tlahuext, O. Muđoz‐Muđiz and H. Torres‐Gómez, Microwave‐Assisted One‐Pot Synthesis of 2‐(Substituted phenyl)‐1 H‐ benzimidazole Derivatives, Synth. Commun., 2007, 37 (17), 2815-2825.

129. R. V. Viesser, L. C. Ducati, C. F. Tormena and J. Autschbach, The halogen effect on the 13 C NMR chemical shift in substituted benzenes, Phys. Chem. Chem. Phys., 2018, 20 (16), 11247-11259.

130. A. S. Al-Bogami, T. S. Saleh, A. E. Mekky and M. R. Shaaban, Microwave assisted regioselective synthesis and 2D-NMR studies of novel azoles and azoloazines utilizing fluorine-containing building Blocks, J. Mol. Struct., 2016, 1121 167-179.

131. W. R. Dolbier Jr, Guide to fluorine NMR for organic chemists, John Wiley & Sons, 2016.

132. V. Sridharan, S. Saravanan, S. Muthusubramanian and S. Sivasubramanian, NMR investigation of hydrogen bonding and 1, 3‐tautomerism in 2‐(2‐ hydroxy‐5‐substituted‐aryl) benzimidazoles, Magnetic Resonance in Chemistry, 2005, 43 (7), 551-556.

133. H. Claussen, I. Dramburg, M. Gastreich, S. Hindle, A. Kamper, B. Kramer,

M. Lilienthal, G. Muller and M. Rarey, User & Technical Reference as Part of LeadIT 2.3, BioSolveIT GmbH, 2017, Augustin, Germany.

134. T. Andoh, K. Ishii, Y. Suzuki, Y. Ikegami, Y. Kusunoki, Y. Takemoto and K. Okada, Characterization of a mammalian mutant with a camptothecin- resistant DNA topoisomerase I, Proc. Natl. Acad. Sci., 1987, 84 (16), 5565- 5569.

135. Y. Fan, J. N. Weinstein, K. Kohn, L. Shi and Y. Pommier, Molecular modeling studies of the DNA− topoisomerase I ternary cleavable complex with camptothecin, J. Med. Chem., 1998, 41 (13), 2216-2226.

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